| 2013 | Design and synthesis of novel series of 5-HT6 receptor ligands having indole, a central aromatic core and 1-amino-4 methyl piperazine as a positive ionizable group | 박혜영 | Article |
| 2021 | Design and Synthesis of TRAP1 Selective Inhibitors: H-Bonding with Asn171 Residue in TRAP1 Increases Paralog Selectivity | 강수성 | Article |
| 2008 | Design and synthesis of truncated 4'-thioadenosine derivatives as potent and selective A3 adenosine receptor antagonists. | 정낙신; 최원준 | Article |
| 2000 | Design and synthesis of α,β-unsaturated carbonyl compounds as potential ACE inhibitors | 박혜영 | Article |
| 2007 | Design, docking, and synthesis of novel indeno[1,2-c]isoquinolines for the development of antitumor agents as topoisomerase I inhibitors | 이상국; 권영주 | Article |
| 2007 | Design, enantiopure synthesis, and biological evaluation of novel ISO-D-2′,3′-dideoxy-3′-fluorothianucleoside derivatives as a bioisostere of lamivudine | 정낙신 | Article |
| 2011 | Design, synthesis and anticancer activity of novel dihydrobenzofuro[4,5-b] [1,8]naphthyridin-6-one derivatives | 정낙신 | Article |
| 2003 | Design, synthesis and binding affinity of 3′-fluoro analogues of Cl-IB-MECA as adenosine A3 receptor ligands | 이승진; 정낙신 | Article |
| 2022 | Design, Synthesis and Biological Evaluation of 1,3,5-Triazine Derivatives Targeting hA(1) and hA(3) Adenosine Receptor | 유진하 | Article |
| 2017 | Design, synthesis and biological evaluation of 1,3-diphenylbenzo[f] [1,7]naphthyrdines | 권영주; 전규연 | Article |
| 2014 | Design, synthesis and biological evaluation of benzyl 2-(1H-imidazole-1-yl) pyrimidine analogues as selective and potent Raf inhibitors | 류재상 | Article |
| 2011 | Design, synthesis and docking study of 5-amino substituted indeno[1,2-c]isoquinolines as novel topoisomerase i inhibitors | 권영주 | Article |
| 2008 | Design, synthesis and evaluation of 2-phenyl-1H-benzo[d]imidazole-4,7-diones as vascular smooth muscle cell proliferation inhibitors | 유충규; 이상국 | Article |
| 2014 | Design, synthesis and systematic evaluation of cytotoxic 3-heteroarylisoquinolinamines as topoisomerases inhibitors | 권영주 | Article |
| 2011 | Design, Synthesis, and Anti-HCV Activity of 2 '-Modified-4 '-selenonucleosides | 정낙신; 최원준; 이혁우 | Meeting Abstract |
| 2007 | Design, synthesis, and anti-tumor activity of 4′-thionucleosides as potent and selective agonists at the human A3 adenosine receptor | 정낙신; 이상국 | Article |
| 2016 | Design, synthesis, and anticancer activity of C8-substituted-4 '-thionucleosides as potential HSP90 inhibitors | 최선 | Article |
| 2007 | Design, synthesis, and anticancer activity of fluorocyclopentenyl-pyrimidines | 정낙신; 이상국 | Meeting Abstract |
| 2005 | Design, synthesis, and anticancer activity of fluorocyclopentenyl-pyrimidines. | 이강만; 정낙신; 이상국; 최원준 | Article |
| 2012 | Design, synthesis, and antitumor evaluation of 2,4,6-triaryl pyridines containing chlorophenyl and phenolic moiety | 권영주 | Article |
